ANGELUCCI, FRANCESCO

ANGELUCCI, FRANCESCO  

Dipartimento di Medicina clinica, sanità pubblica, scienze della vita e dell'ambiente  

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Gold-containing compounds target an apicomplexan Thioredoxin reductase: Disclosing reactivity through structural and functional characterization 1-gen-2026 Gabriele, Federica; Palerma, Marta; Bogard, Jala; Paluzzi, Luca; Zineddu, Stefano; Geri, Andrea; Vitali, Valentina; Massai, Lara; Ardini, Matteo; Bellelli, Andrea; Petukhov, Pavel A.; Ippoliti, Rodolfo; Messori, Luigi; Williams, David L.; Angelucci, Francesco
Unraveling in vitro phase separation and aggregation properties of the structured region of FMRP and the impact of Fragile X syndrome-linked mutations 1-gen-2026 Catalano, Flavia; Bigi, Alessandra; Troilo, Francesca; Gabriele, Federica; Pistoia, Gianluca; Asteriti, Italia A; Angelucci, Francesco; Giardina, Giorgio; Chiti, Fabrizio; Travaglini-Allocatelli, Carlo; Di Matteo, Adele
Unravelling the anti-cancer mechanisms elicited by non-covalent thioredoxin reductase inhibitors for triple negative breast cancer therapy 1-gen-2026 Rullo, Abigail; Flowers, Brenna; Chang, Keacha; Zhang, An; Petukhova, Valentina Z; Harding, Luke; Aboagye, Sammy Y; Bocchetta, Maurizio; Qiu, Wei; Williams, David L; Angelucci, Francesco; Petukhov, Pavel A; Kastrati, Irida
Synthesis of Methoxylated Benzoxanthones as Drug Metabolites of Antischistosomal Schistodiones-A Limited Environmental Risk 1-gen-2026 Cesar-Rodo, Elena; Boilevin, Jeremy; Richard, Jimmy; Ziniel, Peter D; Belorgey, Didier; Maes, Louis; Angelucci, Francesco; Williams, David Lee; Davioud-Charvet, Elisabeth; Lanfranchi, Don Antoine
Heterotropic regulation and negative homotropic cooperativity 1-gen-2026 Morea, Veronica; Angelucci, Francesco; Arnesano, Federica; Pascarella, Gianmarco; Di Micco, Patrizio; Bellelli, Andrea
Targeting Apicomplexan Parasites: Structural and Functional Characterization of Cryptosporidium Thioredoxin Reductase as a Novel Drug Target 1-gen-2025 Gabriele, Federica; Bogard, Jala A.; Palerma, Marta; Ardini, Matteo; Byrne, Margaret E.; Chen, Xian-Ming; Petukhov, Pavel A.; Ippoliti, Rodolfo; Angelucci, Francesco; Williams, David L.
Functional and structural characterization of the human indolethylamine N-methyltransferase through fluorometric, thermal and computational docking analyses 1-gen-2025 Ardini, Matteo; Angelucci, Francesco; Rea, Francesca; Paluzzi, Luca; Gabriele, Federica; Palerma, Marta; Di Leandro, Luana; Ippoliti, Rodolfo; Pitari, Giuseppina
Pleiotropic anti-cancer activities of novel non-covalent thioredoxin reductase inhibitors against triple negative breast cancer 1-gen-2024 Flowers, Brenna; Rullo, Abigail; Zhang, An; Chang, Keacha; Petukhova, Valentina Z.; Aboagye, Sammy Y.; Angelucci, Francesco; Williams, David L.; Kregel, Steven; Petukhov, Pavel A.; Kastrati, Irida
The “Doorstop Pocket” In Thioredoxin Reductases─An Unexpected Druggable Regulator of the Catalytic Machinery 1-gen-2024 Ardini, Matteo; Aboagye, Sammy Y.; Petukhova, Valentina Z.; Kastrati, Irida; Ippoliti, Rodolfo; Thatcher, Gregory R. J.; Petukhov, Pavel A.; Williams, David L.; Angelucci, Francesco
Non-covalent inhibitors of thioredoxin glutathione reductase with schistosomicidal activity in vivo 1-gen-2023 Petukhova, Valentina Z; Aboagye, Sammy Y; Ardini, Matteo; Lullo, Rachel P; Fata, Francesca; Byrne, Margaret E; Gabriele, Federica; Martin, Lucy M; Harding, Luke N M; Gone, Vamshikrishna; Dangi, Bikash; Lantvit, Daniel D; Nikolic, Dejan; Ippoliti, Rodolfo; Effantin, Grégory; Ling, Wai Li; Johnson, Jeremy J; Thatcher, Gregory R J; Angelucci, Francesco; Williams, David L; Petukhov, Pavel A
Recent Advances on Affibody- and DARPin-Conjugated Nanomaterials in Cancer Therapy 1-gen-2023 Gabriele, Federica; Palerma, Marta; Ippoliti, Rodolfo; Angelucci, Francesco; Pitari, Giuseppina; Ardini, Matteo
Truncating variants in the penultimate exon of TGFBR1 escaping nonsense-mediated mRNA decay cause Loeys-Dietz syndrome 1-gen-2023 Fortugno, Paola; Monetta, Rosanna; Cinquina, Valeria; Rigon, Chiara; Boaretto, Francesca; De Luca, Chiara; Zoppi, Nicoletta; Di Leandro, Luana; De Domenico, Emanuela; Di Daniele, Arianna; Ippoliti, Rodolfo; Angelucci, Francesco; Di Cesare, Ernesto; De Paulis, Ruggero; Salviati, Leonardo; Colombi, Marina; Brancati, Francesco; Ritelli, Marco
Molecular dynamics simulations and kinetic measurements provide insights into the structural requirements of substrate size-dependent specificity of oligogalacturonide oxidase 1 (OGOX1) 1-gen-2023 Frezzini, Mario; Scortica, Anna; Capone, Matteo; Narzi, Daniele; Benedetti, Manuel; Angelucci, Francesco; Mattei, Benedetta; Guidoni, Leonardo
Bio-Tailored Sensing at the Nanoscale: Biochemical Aspects and Applications 1-gen-2023 Fata, Francesca; Gabriele, Federica; Angelucci, Francesco; Ippoliti, Rodolfo; Di Leandro, Luana; Giansanti, Francesco; Ardini, Matteo
COMPOUNDS AND METHODS FOR THE TREATMENT OF DISEASES ASSOCIATED WITH PARASITIC WORMS 1-gen-2022 Petukhov, Pavel; Petukhov, Valentina; Williams, David; Angelucci, Francesco; Aboagye, Samuel; Ardini, Matteo
First non-covalent inhibitors of thioredoxin glutathione reductase with schistosomicidal activity in vivo 1-gen-2022 Petukhova, Valentina; Aboagye, Samuel; Ardini, Matteo; Lullo, Rachel; Byrne, Margaret; Martin, Lucy; Fata, Francesca; Gabriele, Federica; Ippoliti, Rodolfo; Ling, Wai Li; Effantin, Grégory; Harding, Luke; Nikolic, Dejan; Lantvit, Daniel; Dangi, Bikash; Gone, Vamshikrishna; Johnson, Jeremy; Thatcher, Gregory; Angelucci, Francesco; Williams, David; Petukhov, Pavel
Tuning the Sensing Properties of N and S Co-Doped Carbon Dots for Colorimetric Detection of Copper and Cobalt in Water 1-gen-2022 Bisauriya, R.; Antonaroli, S.; Ardini, M.; Angelucci, F.; Ricci, A.; Pizzoferrato, R.
Characterization of two 1,3-β-glucan-modifying enzymes from Penicillium sumatraense reveals new insights into 1,3-β-glucan metabolism of fungal saprotrophs 1-gen-2022 Scafati, Valentina; Troilo, Francesca; Ponziani, Sara; Giovannoni, Moira; Scortica, Anna; Pontiggia, Daniela; Angelucci, Francesco; Di Matteo, Adele; Mattei, Benedetta; Benedetti, Manuel
RIPK4 regulates cell-cell adhesion in epidermal development and homeostasis 1-gen-2022 Fortugno, Paola; Monetta, Rosanna; Belli, Manuel; Botti, Elisabetta; Angelucci, Francesco; Palmerini, Maria Grazia; Annarita, Nottola Stefania; De Luca, Chiara; Ceccarini, Marina; Salvatore, Marco; Bianchi, Luca; Macioce, Pompeo; Teson, Massimo; Ricci, Francesco; Network, Italian Undiagnosed Diseases; Macchiarelli, Guido; Didona, Biagio; Costanzo, Antonio; Castiglia, Daniele; Brancati, Francesco
Structural Basis of Sequential and Concerted Cooperativity 1-gen-2022 Morea, Veronica; Angelucci, Francesco; Tame, Jeremy R. H.; Di Cera, Enrico Di; Bellelli, Andrea